CAS No.:19237-84-4
Name: Prazosin hydrochloride
Details Introduction
TOXICITY DATA with REFERENCE:
Organism | Test Type | Route | Reported Dose (Normalized Dose) | Effect | Source |
---|---|---|---|---|---|
dog | LD50 | oral | > 700mg/kg (700mg/kg) | GASTROINTESTINAL: CHANGES IN STRUCTURE OR FUNCTION OF SALIVARY GLANDS GASTROINTESTINAL: NAUSEA OR VOMITING KIDNEY, URETER, AND BLADDER: OTHER CHANGES |
Oyo Yakuri. Pharmacometrics. Vol. 17, Pg. 39, 1979. |
human | TDLo | oral | 285ug/kg (0.285mg/kg) | VASCULAR: BP LOWERING NOT CHARACTERIZED IN AUTONOMIC SECTION | JAMA, Journal of the American Medical Association. Vol. 238, Pg. 157, 1977. |
man | TDLo | oral | 1714ug/kg (1.714mg/kg) | BEHAVIORAL: COMA LUNGS, THORAX, OR RESPIRATION: DYSPNEA |
Human Toxicology. Vol. 4, Pg. 53, 1985 |
mouse | LD50 | intraperitoneal | 60mg/kg (60mg/kg) | BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY) GASTROINTESTINAL: "HYPERMOTILITY, DIARRHEA" BEHAVIORAL: ATAXIA |
Oyo Yakuri. Pharmacometrics. Vol. 17, Pg. 39, 1979. |
mouse | LD50 | intravenous | 92mg/kg (92mg/kg) | BEHAVIORAL: CONVULSIONS OR EFFECT ON SEIZURE THRESHOLD LUNGS, THORAX, OR RESPIRATION: DYSPNEA BEHAVIORAL: ATAXIA |
New Cardiovascular Drugs. Vol. 4, Pg. 1, 1986. |
mouse | LD50 | oral | 5gm/kg (5000mg/kg) | Medicamentos de Actualidad. Vol. 11, Pg. 64, 1975. | |
mouse | LD50 | subcutaneous | 3100mg/kg (3100mg/kg) | BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY) LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION BEHAVIORAL: ATAXIA |
Oyo Yakuri. Pharmacometrics. Vol. 17, Pg. 39, 1979. |
rat | LD50 | intraperitoneal | 102mg/kg (102mg/kg) | SENSE ORGANS AND SPECIAL SENSES: LACRIMATION: EYE LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY) |
Oyo Yakuri. Pharmacometrics. Vol. 17, Pg. 39, 1979. |
rat | LD50 | intravenous | 73mg/kg (73mg/kg) | BEHAVIORAL: CONVULSIONS OR EFFECT ON SEIZURE THRESHOLD BEHAVIORAL: ATAXIA LUNGS, THORAX, OR RESPIRATION: DYSPNEA |
New Cardiovascular Drugs. Vol. 4, Pg. 1, 1986. |
rat | LD50 | oral | 1950mg/kg (1950mg/kg) | GASTROINTESTINAL: CHANGES IN STRUCTURE OR FUNCTION OF SALIVARY GLANDS GASTROINTESTINAL: NAUSEA OR VOMITING KIDNEY, URETER, AND BLADDER: OTHER CHANGES |
Oyo Yakuri. Pharmacometrics. Vol. 17, Pg. 39, 1979. |
rat | LD50 | subcutaneous | 3750mg/kg (3750mg/kg) | SENSE ORGANS AND SPECIAL SENSES: LACRIMATION: EYE BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY) LUNGS, THORAX, OR RESPIRATION: RESPIRATORY DEPRESSION |
Oyo Yakuri. Pharmacometrics. Vol. 17, Pg. 39, 1979. |
women | TDLo | oral | 10ug/kg (0.01mg/kg) | BEHAVIORAL: COMA VASCULAR: BP LOWERING NOT CHARACTERIZED IN AUTONOMIC SECTION SKIN AND APPENDAGES (SKIN): SWEATING: OTHER |
Drug Intelligence and Clinical Pharmacy. Vol. 21, Pg. 723, 1987. |
women | TDLo | oral | 13mg/kg/6W-I (13mg/kg) | BRAIN AND COVERINGS: ENCEPHALITIS BEHAVIORAL: SOMNOLENCE (GENERAL DEPRESSED ACTIVITY) BEHAVIORAL: TOXIC PSYCHOSIS |
British Medical Journal. Vol. 293, Pg. 1347, 1986. |
Consensus Reports:
SAFETY PROFILE:
Safety Information of Prazosin hydrochloride (CAS NO.19237-84-4):
Hazard Codes: Xn
Risk Statements: 22-36/37/38-62
22: Harmful if swallowed
36: Irritating to the eyes
37: Irritating to the respiratory system
38: Irritating to the skin
Possible risk of impaired fertility
Safety Statements: 28-36
28: After contact with skin, wash immediately with plenty of ... (to be specified by the manufacturer)
36: Wear suitable protective clothing
Standards and Recommendations:
Analytical Methods:
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