CAS No.:33396-37-1
Name: Meproscillarin
Details Introduction
TOXICITY DATA with REFERENCE:
| Organism | Test Type | Route | Reported Dose (Normalized Dose) | Effect | Source |
|---|---|---|---|---|---|
| cat | LDLo | intravenous | 137ug/kg (0.137mg/kg) | Arzneimittel-Forschung. Drug Research. Vol. 28, Pg. 495, 1978. | |
| guinea pig | LDLo | intravenous | 678ug/kg (0.678mg/kg) | Arzneimittel-Forschung. Drug Research. Vol. 28, Pg. 495, 1978. | |
| mouse | LD50 | intravenous | 2800ug/kg (2.8mg/kg) | BEHAVIORAL: ALTERED SLEEP TIME (INCLUDING CHANGE IN RIGHTING REFLEX) BEHAVIORAL: TREMOR BEHAVIORAL: CONVULSIONS OR EFFECT ON SEIZURE THRESHOLD |
Arzneimittel-Forschung. Drug Research. Vol. 28, Pg. 506, 1978. |
| mouse | LD50 | oral | 12500ug/kg (12.5mg/kg) | BEHAVIORAL: ALTERED SLEEP TIME (INCLUDING CHANGE IN RIGHTING REFLEX) BEHAVIORAL: TREMOR BEHAVIORAL: CONVULSIONS OR EFFECT ON SEIZURE THRESHOLD |
Arzneimittel-Forschung. Drug Research. Vol. 28, Pg. 506, 1978. |
| rat | LD50 | intravenous | 5800ug/kg (5.8mg/kg) | BEHAVIORAL: ALTERED SLEEP TIME (INCLUDING CHANGE IN RIGHTING REFLEX) BEHAVIORAL: TREMOR BEHAVIORAL: CONVULSIONS OR EFFECT ON SEIZURE THRESHOLD |
Arzneimittel-Forschung. Drug Research. Vol. 28, Pg. 506, 1978. |
| rat | LD50 | oral | 79mg/kg (79mg/kg) | BEHAVIORAL: ALTERED SLEEP TIME (INCLUDING CHANGE IN RIGHTING REFLEX) BEHAVIORAL: TREMOR BEHAVIORAL: CONVULSIONS OR EFFECT ON SEIZURE THRESHOLD |
Arzneimittel-Forschung. Drug Research. Vol. 28, Pg. 506, 1978. |
Consensus Reports:
SAFETY PROFILE:
Poison by ingestion and intravenous routes. Experimental reproductive effects. When Meproscillarin (CAS NO.33396-37-1) is heated to decomposition, it emits acrid smoke and irritating fumes.
Standards and Recommendations:
Analytical Methods:
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